Esters of Phosphorus Oxy Acids as Alkylating Agents. IV.N-Alkylation of Imidazole and Its Analogs with Alkyl Esters of Phosphonic and Phosphinic Acids
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LONG-ACTING CONTRACEPTIVE AGENTS: TESTOSTERONE ESTERS OF CYCLOALKYLCARBOXYLIC ACIDS
The synthesis of twenty five esters of testosterone (17β -hydroxyandrost- 4-en-3-one) is described. All esters are derivatives of cycloalkycarboxylic acids. Some of the esters possess α- , β -and/or & - substitution in the ester side-chain. The work was undertaken in order to evaluate long-acting male antifertility effect of such esters. Most of the compounds, especially compound No.1, wer...
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the synthesis of twenty five esters of testosterone (17β -hydroxyandrost- 4-en-3-one) is described. all esters are derivatives of cycloalkycarboxylic acids. some of the esters possess α- , β -and/or & - substitution in the ester side-chain. the work was undertaken in order to evaluate long-acting male antifertility effect of such esters. most of the compounds, especially compound no.1, were fou...
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ژورنال
عنوان ژورنال: Bulletin of the Chemical Society of Japan
سال: 1976
ISSN: 0009-2673,1348-0634
DOI: 10.1246/bcsj.49.283